Drugs Information:
Ponesimod
Basic Information
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| ID | DDInter2039 | |
| Drug Type | small molecule | |
| Molecular Formula | C23H25ClN2O4S | |
| Molecular Weight | 460.970 | |
| CAS Number | 854107-55-4 | |
| Description | Ponesimod is a selective sphingosine 1-phosphate receptor 1 modulator indicated in the treatment of relapsing forms of multiple sclerosis in adults.[A232079,L32709] Ponesimod was developed out of a need for a more selective modulator of sphingosine 1-phosphate receptor 1 than [fingolimod].[A232079] Fingolimod's activity at sphingosine 1-phosphate receptor 3 was suspected to be responsible for a portion of it's adverse effects, and so more selective modulators were developed.[A232079] Ponesimod was granted FDA approval on 18 March 2021.[L32709] | |
| ATC Classification | L04AA50 | |
| IUPAC Name | (2Z,5Z)-5-({3-chloro-4-[(2R)-2,3-dihydroxypropoxy]phenyl}methylidene)-3-(2-methylphenyl)-2-(propylimino)-1,3-thiazolidin-4-one | |
| InChI | LPAUOXUZGSBGDU-STDDISTJSA-N | |
| Canonical SMILES | CCC\N=C1/S\C(=C/C2=CC=C(OC[C@H](O)CO)C(Cl)=C2)C(=O)N1C1=CC=CC=C1C | |
| Useful Links | DrugBank PubChem Substance ChemSpider BindingDB Wikipedia ChEMBL ZINC | |
Interactions with
Ponesimod
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Interactions with foods
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Interactions with compound preparation
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