Drugs Information:
Rotigotine
Basic Information
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ID | DDInter1624 | |
Drug Type | small molecule | |
Molecular Formula | C19H25NOS | |
Molecular Weight | 315.480 | |
CAS Number | 99755-59-6 | |
Description | Rotigotine (Neupro) is a non-ergoline dopamine agonist indicated for the treatment of Parkinson's disease (PD) and restless legs syndrome (RLS) in Europe and the United States. It is formulated as a once-daily transdermal patch which provides a slow and constant supply of the drug over the course of 24 hours. Like other dopamine agonists, rotigotine has been shown to possess antidepressant effects and may be useful in the treatment of depression as well. Rotigotine was developed by Aderis Pharmaceuticals. In 1998 Aderis licensed worldwide development and commercialization rights to Schwarz Pharma of Germany. It was approved by the European Medicines Agency in 2006 and by the FDA in 2007. However, all Neupro patches in the United States and some of Europe were recalled in 2008 due to delivery mechanism issues. Rotigotine has been authorized as a treatment for RLS since August 2008. | |
ATC Classification | N04BC09 | |
IUPAC Name | (6S)-6-{propyl[2-(thiophen-2-yl)ethyl]amino}-5,6,7,8-tetrahydronaphthalen-1-ol | |
InChI | KFQYTPMOWPVWEJ-INIZCTEOSA-N | |
Canonical SMILES | CCCN(CCC1=CC=CS1)[C@H]1CCC2=C(O)C=CC=C2C1 | |
Useful Links | DrugBank ChEBI PubChem Substance KEGG Drug ChemSpider BindingDB PharmGKB Guide to Pharmacology Wikipedia ChEMBL ZINC |
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Rotigotine
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