Drugs Information:
Perindopril
Basic Information
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ID | DDInter1431 | |
Drug Type | small molecule | |
Molecular Formula | C19H32N2O5 | |
Molecular Weight | 368.468 | |
CAS Number | 82834-16-0 | |
Description | Perindopril is a nonsulfhydryl prodrug that belongs to the angiotensin-converting enzyme (ACE) inhibitor class of medications. It is rapidly metabolized in the liver to perindoprilat, its active metabolite, following oral administration. Perindoprilat is a potent, competitive inhibitor of ACE, the enzyme responsible for the conversion of angiotensin I (ATI) to angiotensin II (ATII). ATII regulates blood pressure and is a key component of the renin-angiotensin-aldosterone system (RAAS). Perindopril may be used to treat mild to moderate essential hypertension, mild to moderate congestive heart failure, and to reduce the cardiovascular risk of individuals with hypertension or post-myocardial infarction and stable coronary disease. | |
ATC Classification | C09BX01 C09BA04 C10BX11 C10BX13 C09AA04 C09BX02 C10BX12 C09BB04 C10BX15 C10BX14 C09BX04 | |
IUPAC Name | (2S,3aS,7aS)-1-[(2S)-2-{[(2S)-1-ethoxy-1-oxopentan-2-yl]amino}propanoyl]-octahydro-1H-indole-2-carboxylic acid | |
InChI | IPVQLZZIHOAWMC-QXKUPLGCSA-N | |
Canonical SMILES | [H][C@]12C[C@H](N(C(=O)[C@H](C)N[C@@H](CCC)C(=O)OCC)[C@@]1([H])CCCC2)C(O)=O | |
Useful Links | DrugBank ChEBI PubChem Substance KEGG Compound KEGG Drug ChemSpider BindingDB PharmGKB Therapeutic Targets Database Wikipedia ChEMBL ZINC |
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Perindopril
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