Drugs Information:
Apixaban
Basic Information
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ID | DDInter108 | |
Drug Type | small molecule | |
Molecular Formula | C25H25N5O4 | |
Molecular Weight | 459.497 | |
CAS Number | 503612-47-3 | |
Description | Apixaban is an oral, direct, and highly selective factor Xa (FXa) inhibitor of both free and bound FXa, as well as prothrombinase, independent of antithrombin III for the prevention and treatment of thromboembolic diseases[Label,A6897]. It is marketed under the name Eliquis[Label,L6043]. Apixaban was approved by the FDA on December 28, 2012[L6043]. | |
ATC Classification | B01AF02 | |
IUPAC Name | 1-(4-methoxyphenyl)-7-oxo-6-[4-(2-oxopiperidin-1-yl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridine-3-carboxamide | |
InChI | QNZCBYKSOIHPEH-UHFFFAOYSA-N | |
Canonical SMILES | COC1=CC=C(C=C1)N1N=C(C(N)=O)C2=C1C(=O)N(CC2)C1=CC=C(C=C1)N1CCCCC1=O | |
Useful Links | DrugBank ChEBI PubChem Substance KEGG Drug ChemSpider BindingDB PharmGKB Wikipedia ChEMBL ZINC |
Interactions with
Apixaban
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Interactions with compound preparation
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